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Synthesis and Superpotent Anticancer Activity of Tubulysins Carrying Non-hydrolysable N-Substituents on Tubuvaline

dc.contributor.authorSani, Monica
dc.contributor.authorLazzari, Paolo
dc.contributor.authorFolini, Marco
dc.contributor.authorSpiga, Marco
dc.contributor.authorZuco, Valentina
dc.contributor.authorDe Cesare, Michelandrea
dc.contributor.authorManca, Ilaria
dc.contributor.authorDall'Angelo, Sergio
dc.contributor.authorFrigerio, Massimo
dc.contributor.authorUsai, Igor
dc.contributor.authorTesta, Andrea
dc.contributor.authorZaffaroni, Nadia
dc.contributor.authorZanda, Matteo
dc.contributor.institutionUniversity of Aberdeen.Medical Sciencesen
dc.contributor.institutionUniversity of Aberdeen.Medical Sciences - Cardiovascular Groupen
dc.date.accessioned2018-04-12T23:02:53Z
dc.date.available2018-04-12T23:02:53Z
dc.date.embargoedUntil2018-04-12
dc.date.issued2017-04-27
dc.descriptionWe thank Regione Autonoma della Sardegna RAS (Italy) for economic support by covering in part the costs of this research. I.U. acknowledges RAS for his fellowship (for grant numbers see the Supporting Information)en
dc.description.statusPeer revieweden
dc.format.extent9
dc.format.extent437107
dc.identifier95760605
dc.identifierd1d8d2a8-af22-4534-95a5-c33da18d9dd5
dc.identifier85017578993
dc.identifier.citationSani, M, Lazzari, P, Folini, M, Spiga, M, Zuco, V, De Cesare, M, Manca, I, Dall'Angelo, S, Frigerio, M, Usai, I, Testa, A, Zaffaroni, N & Zanda, M 2017, 'Synthesis and Superpotent Anticancer Activity of Tubulysins Carrying Non-hydrolysable N-Substituents on Tubuvaline', Chemistry : a European Journal, vol. 23, no. 24, pp. 5842-5850. https://doi.org/10.1002/chem.201700874en
dc.identifier.doi10.1002/chem.201700874
dc.identifier.iss24en
dc.identifier.issn0947-6539
dc.identifier.otherORCID: /0000-0001-9377-0474/work/176747534
dc.identifier.urihttp://hdl.handle.net/2164/10324
dc.identifier.vol23en
dc.language.isoeng
dc.relation.ispartofChemistry : a European Journalen
dc.subjectSDG 3 - Good Health and Well-beingen
dc.subjecttubulysinsen
dc.subjectantitumoren
dc.subjectaza-Michaelen
dc.subjectin vitro testsen
dc.subjectin vivo testsen
dc.subjectQD Chemistryen
dc.subject.lccQDen
dc.titleSynthesis and Superpotent Anticancer Activity of Tubulysins Carrying Non-hydrolysable N-Substituents on Tubuvalineen
dc.typeJournal articleen

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