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Synthesis and Biological Evaluation of Indole-2-Carboxamides with Potent Apoptotic Antiproliferative Activity as EGFR/CDK2 Dual Inhibitors

dc.contributor.authorAl-Wahaibi, Lamya H.
dc.contributor.authorMostafa, Yaser A.
dc.contributor.authorAbdelrahman, Mostafa H.
dc.contributor.authorEl-Bahrawy, Ali H.
dc.contributor.authorTrembleau, Laurent
dc.contributor.authorYoussif, Bahaa G.M.
dc.contributor.institutionUniversity of Aberdeen.Chemistryen
dc.date.accessioned2023-04-25T12:19:01Z
dc.date.available2023-04-25T12:19:01Z
dc.date.issued2022-08-16
dc.descriptionFunding Information: This work was funded by Princess Nourah bint Abdulrahman University Researchers Supporting Project Number (PNURSP2022R3), Princess Nourah bint Abdulrahman University, Riyadh, Saudi Arabia.en
dc.description.statusPeer revieweden
dc.format.extent17
dc.format.extent4037582
dc.identifier219534384
dc.identifierb3f237d6-bbbf-4738-bb94-6141e57eeabe
dc.identifier85137348607
dc.identifier36015154
dc.identifier.citationAl-Wahaibi, L H, Mostafa, Y A, Abdelrahman, M H, El-Bahrawy, A H, Trembleau, L & Youssif, B G M 2022, 'Synthesis and Biological Evaluation of Indole-2-Carboxamides with Potent Apoptotic Antiproliferative Activity as EGFR/CDK2 Dual Inhibitors', Pharmaceuticals, vol. 15, no. 8, 1006. https://doi.org/10.3390/ph15081006en
dc.identifier.doi10.3390/ph15081006
dc.identifier.iss8en
dc.identifier.issn1424-8247
dc.identifier.otherORCID: /0000-0001-6376-9077/work/133803283
dc.identifier.urihttps://hdl.handle.net/2164/20556
dc.identifier.urlhttp://www.scopus.com/inward/record.url?scp=85137348607&partnerID=8YFLogxKen
dc.identifier.vol15en
dc.language.isoeng
dc.relation.ispartofPharmaceuticalsen
dc.subjectSDG 3 - Good Health and Well-beingen
dc.subjectantiproliferativeen
dc.subjectapoptosisen
dc.subjectcarboxamideen
dc.subjectindoleen
dc.subjectmulti-targeten
dc.subjectQD Chemistryen
dc.subjectMolecular Medicineen
dc.subjectPharmaceutical Scienceen
dc.subjectDrug Discoveryen
dc.subject.lccQDen
dc.titleSynthesis and Biological Evaluation of Indole-2-Carboxamides with Potent Apoptotic Antiproliferative Activity as EGFR/CDK2 Dual Inhibitorsen
dc.typeJournal articleen

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