Sani, MonicaLazzari, PaoloFolini, MarcoSpiga, MarcoZuco, ValentinaDe Cesare, MichelandreaManca, IlariaDall'Angelo, SergioFrigerio, MassimoUsai, IgorTesta, AndreaZaffaroni, NadiaZanda, Matteo2018-04-122018-04-122017-04-27Sani, M, Lazzari, P, Folini, M, Spiga, M, Zuco, V, De Cesare, M, Manca, I, Dall'Angelo, S, Frigerio, M, Usai, I, Testa, A, Zaffaroni, N & Zanda, M 2017, 'Synthesis and Superpotent Anticancer Activity of Tubulysins Carrying Non-hydrolysable N-Substituents on Tubuvaline', Chemistry : a European Journal, vol. 23, no. 24, pp. 5842-5850. https://doi.org/10.1002/chem.2017008740947-6539ORCID: /0000-0001-9377-0474/work/176747534http://hdl.handle.net/2164/10324We thank Regione Autonoma della Sardegna RAS (Italy) for economic support by covering in part the costs of this research. I.U. acknowledges RAS for his fellowship (for grant numbers see the Supporting Information)9437107engSDG 3 - Good Health and Well-beingtubulysinsantitumoraza-Michaelin vitro testsin vivo testsQD ChemistryQDJournal article10.1002/chem.2017008742324